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. 2012 Apr;31(4):178–184. doi: 10.5732/cjc.011.10290

Table 1. The half maximal inhibition concentration (IC50) values of niclosamide in some tumor cell lines and normal cells.

Tumor type Cell line IC50 (µmol/L) Reference
Leukemia
 Acute myeloid leukemia U937 0.41 [2]
OCI-AML3 0.79 [2]
HL-60 0.48 [2]
Molm13 0.72 [2]
MV4-11 1.0 [2]
Solid tumor
 Prostrate cancer Du145 0.7 [5]
PC3 11.7±2.3 [5]
 Colorectal cancer HT29 7.2±1.2 [5]
HCT116 2.2 [4]
 Cervical carcinoma HeLa 0.25±0.07 [5]
 Lung adenocarcinoma A549 3.0±0.2 [5]
 Epithelial carcinoma A431 8.8±0.9 [5]
Normal cell
MEF 4.54 [2]
NHFB 5.78 [2]
Bone marrow 9.00±4.87 [2]