Evaluation
of NHS carbamates as serine hydrolase inhibitors. (A) Structures of
representative members of NHS carbamate library. (B) In vitro evaluation
of NHS carbamates as serine hydrolase inhibitors in mouse brain (membrane)
proteomes showing inhibition of multiple serine hydrolases including
MAGL, FAAH, ABHD6, LYPLA1/2, and APEH (enzyme identities were assigned
based on gel migration patterns consistent with previous studies3b,3c,29). See Figure
S1 for full compound list and ABPP gel profiles.