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. Author manuscript; available in PMC: 2014 Jun 25.
Published in final edited form as: Biochemistry. 2013 Jun 11;52(25):4391–4398. doi: 10.1021/bi400264d

Table 2.

Inhibition and Binding Constants of 2-Aminothiazoles for CeUGMa

% Inhibition at 10 μM IC50 (μM) Ki (μM)
3 83 ± 6 3.3 ± 1.1 1.3 ± 0.4
4 95 ± 1 1.8 ± 1.2 0.7 ± 0.5
5 16 ± 3 n/d n/d
a

n/d represents not determined. Ki values were calculated using the Cheng-Prusoff equation.68