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. Author manuscript; available in PMC: 2014 May 28.
Published in final edited form as: J Control Release. 2013 Mar 6;168(1):88–102. doi: 10.1016/j.jconrel.2013.02.020

Table 3. In vivo PDT studies reported on nanoparticle-based photosensitizer formulations.

Photosensitizer NP Vehicle Targeting Motif Cell Type Ref.
Porphyrin derivatives (hematoporphyrin, porfimer sodium etc.) PLGA nanoparticles N/A (Passive) SW480 (human colon cancer) [41]
Polyacrylamide nanoparticles F3 peptide 9L (orthotopic rat glioma) [46, 112]
Magnetic chitosan nanoparticles N/A (Passive) SW480 (xenograft human colon) [35]
Silica nanoparticles N/A (Passive) HeLa (human colon cancer)
HCT 116 (human colon cancer)
A549 (human lung cancer)
[37, 38]
Chlorin derivatives (chlorin e6, mTHPC, pheophorbide etc) Human serum albumin nanoparticles N/A (Passive) HT-29 (human colon cancer) [99]
Chitosan nanoparticles N/A (Passive) HT-29 (human colon cancer) [98]
Iron oxide nanoparticles N/A (Passive) MGC-803 (human gastric cancer) [63]
NaYF4:Yb,Er/NaGdF4 nanoparticles N/A (Passive) U87MG (human glioma) [64]
Hyaluronic acid nanoparticles Hyaluronic acid targeted to CD44 HT-29 (human colon cancer) [61]
PLGA nanoparticles N/A (Passive) Rhabdomyosarcoma (orthotopic) [101]
Polyacrylamide nanoparticles N/A (Passive) Colon-26 (murine colon cancer) [102, 111]
Phthalocyanine derivatives (zinc (II) phthalocyanine, silicon phthalocyanine 4 etc.) Mesoporous silica nanoparticles N/A (Passive) H22 (human hepatoma) [108]
Dendrimers N/A (Passive) A549 (human lung cancer) [109]
Gold nanoparticles EGF Gli36 (orthotopic human glioma) [73]
Indocyanine green Calcium phosphosilicate Anti-CD117 antibody 32D-p210-GFP (orthotopic murine chronic myeloid leukemia) [84]
Methylene blue Phosphonate-terminated silica nanoparticles N/A (Passive) HeLa (human cervical cancer) [91]