Table 2.
Pharmacological inhibition of FAAH inhibition and properties of psychostimulants.
| FAAH inhibitors | Drug | Animal | Outcome | Effects | Reference |
|---|---|---|---|---|---|
| AM404 | Cocaine | Rat | Drug-induced lowering of brain reward/self-stimulation threshold | Impaired | Vlachou et al. (252) |
| Drug-induced acute hyperlocomotion | Attenuated | Vlachou et al. (252) | |||
| URB597 | Cocaine | Monkey | SA – effect of agonist after drug-taking extinction | No effect | Justinova et al. (260) |
| SA – drug-taking behavior | No change | Justinova et al. (260) | |||
| Rat | Cocaine-induced increase in VTA DA activity | Preserved | Luchicchi et al. (259) | ||
| Cocaine-induced alterations in firing of NAc shell spiny neurons | Attenuated | Luchicchi et al. (259) | |||
| URB597, PMSF | Cocaine | Rat | SA – drug-seeking responses/intake | No change | Adamczyk et al. (261) |
| SA – drug-induced reinstatement | Attenuated | Adamczyk et al. (261) | |||
| SA – cue-induced reinstatement | Attenuated | Adamczyk et al. (261) |