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. Author manuscript; available in PMC: 2014 Sep 1.
Published in final edited form as: Bioorg Med Chem. 2013 Jun 15;21(17):5373–5382. doi: 10.1016/j.bmc.2013.06.012

Figure 2.

Figure 2

JTE-013 inhibition of agonists in the S1PR2-CRE-bla assay. Dose response of S1P (A) or CYM5520 (B) on S1PR2- Cre-bla CHO cells was challenged with increasing concentrations of JTE-013 (● DMSO control, ■ 10 nM JTE-013, ▲ 30 nM JTE-013, ▼ 90 nM JTE-013).