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. Author manuscript; available in PMC: 2014 Sep 28.
Published in final edited form as: Org Biomol Chem. 2013 Sep 28;11(36):6036–6046. doi: 10.1039/c3ob40900g

Table 3.

Array of thiomorpholinone-tetrazole derivatives 20

graphic file with name nihms515809t35.jpg
R1 R2 Product Ugi
(%)		 Final Steps*
(%)
graphic file with name nihms515809t36.jpg graphic file with name nihms515809t37.jpg 20a 78 88
graphic file with name nihms515809t38.jpg graphic file with name nihms515809t39.jpg 20b 61 66
graphic file with name nihms515809t40.jpg graphic file with name nihms515809t41.jpg 20c 42 22
graphic file with name nihms515809t42.jpg graphic file with name nihms515809t43.jpg 20d 86 73
graphic file with name nihms515809t44.jpg graphic file with name nihms515809t45.jpg 20e 61 96
*

Basic hydrolysis and SOCl2 activation