Table 2.
Docetaxel pharmacokinetic parameters of 9%-NP and 20%-NP
Specimen | Parameter | Formulation | |
---|---|---|---|
9%-NP | 20%-NP | ||
Plasma | AUC (ng/mL h) | 95,692 (0–72 h) | 82,743 (0–72 h) |
Cmax (ng/mL) | 19,583 ± 7,997 | 26,753 ± 5,603 | |
CL (mL/h/kg) | 105 | 121 | |
Vd (mL/kg) | 943 | 1278 | |
T1/2 (h) | 6.6 | 7.4 | |
Tumor | AUC (ng/mL h) | 99,586 (0–168 h) | 71,848 (0–168 h) |
Cmax (ng/mL) | 1,199 ± 1,115 | 1038 ± 366 | |
Liver | AUC (ng/mL h) | 1,080,179 (0–168 h) | 1,513,225 (0–168 h) |
Cmax (ng/mL) | 16,359 ± 11,681 | 19,274 ± 10,838 | |
Spleen | AUC (ng/mL h) | 5,282,385 (0–168 h) | 6,934,196 (0–168 h) |
Cmax (ng/mL) | 44,294 ± 26,239 | 73,061 ± 10,855 | |
Lung | AUC (ng/mL h) | 165,962 (0–168 h) | 258,766 (0–168 h) |
Cmax (ng/mL) | 17,218 ± 6,347 | 20,200 ± 2,861 |