Table 10.
Fragment-based PanC Inhibitors
| compound | KD (μM) |
|---|---|
153
|
1100 |
154
|
500 |
155
|
500 |
156
|
210 |
157
|
29.0 |
158
|
1.5 |
159
|
1.8 |
Fragment-based PanC Inhibitors
| compound | KD (μM) |
|---|---|
153
|
1100 |
154
|
500 |
155
|
500 |
156
|
210 |
157
|
29.0 |
158
|
1.5 |
159
|
1.8 |