Table 2.
MenE Inhibitors
| compound | IC50 (Kii), μM |
|---|---|
29
|
38 ± 3 |
30
|
34 ± 3 |
31
|
5.7 ± 0.7 |
32
|
> 200 |
33
|
(5.4 ± 0.8)a |
Kii value: Kii(ATP) = 5.2 ± 0.8 μM, Kii(OSB) = 5.6 ± 0.8 μM
MenE Inhibitors
| compound | IC50 (Kii), μM |
|---|---|
29
|
38 ± 3 |
30
|
34 ± 3 |
31
|
5.7 ± 0.7 |
32
|
> 200 |
33
|
(5.4 ± 0.8)a |
Kii value: Kii(ATP) = 5.2 ± 0.8 μM, Kii(OSB) = 5.6 ± 0.8 μM