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. 2010 Aug 13;68(4):709–720. doi: 10.1007/s00018-010-0480-x

Table 1.

Cytotoxicity of F- and Cl-amidine

Cell line Cl-amidine F-amidine
Approximate EC50 Survival (%)a Approximate EC50 Survival (%)a
HL-60 0.25 38 0.5 79
HL-60 granulocytes 100 100
MCF7 0.05 50 0.5 77
HT-29 1 59 1 91
NIH 3T3 100 100

aBased on cell viability at the maximum agent concentration tested