Skip to main content
. Author manuscript; available in PMC: 2014 Sep 1.
Published in final edited form as: Bioorg Med Chem. 2013 Jun 26;21(17):10.1016/j.bmc.2013.06.046. doi: 10.1016/j.bmc.2013.06.046

Scheme 1.

Scheme 1

Reagents and conditions: (a) NaH, toluene, reflux; (b) 3,4-methylenedioxy aniline, toluene, reflux; (c) PPA, 100–110 °C.