Table 5.
Log KD values obtained from [3H]-CGP 12177 whole-cell binding studies in CHO cells stably expressing either the human β1-adrenoceptor or the human β2-adrenoceptor
| ICI 118551 | ||||||
|---|---|---|---|---|---|---|
| CGP 20712A | n | Log KD | n | Retigabine | n | |
| β1 | −8.98 ± 0.08 | 4 | −6.76 ± 0.03 | 4 | No binding | 4 |
| β2 | −5.88 ± 0.02 | 4 | −9.38 ± 0.04 | 4 | No binding | 4 |
Values are mean ± SEM for n separate experiments (Experiment 3).