Table 1.
Cytotoxicity levels (IC50) of rGel, cG-L and rG-L in various cancer cell lines (CT 26, LS174T, 9L and PC-3).
Samples | CT 26a | LS174Ta | 9La | PC-3a |
---|---|---|---|---|
rGel | 1630 ± 510 | 5870 ± 1030 | 3100 ± 420 | 3430 ± 1140 |
cG-L | 37.3 ± 15.7*** | 123.1 ± 26.9*** | 1062 ± 22.7*** | 57.8 ± 23.4** |
rG-L | 79.1 ± 21.4*** | 67.8 ± 13.7*** | 61.3 ± 12.2*** | 83.6 ± 28.3** |
IC50 values are displayed as nM.
P < 0.001
P < 0.0001.
For all experiments, N=3. (rGel: recombinant gelonin, cG-L: gelonin-LMWP chemical conjugate, rG-L: recombinant gelonin-LMWP chimera)