Table 7.
PLS statistics | CoMFA | CoMSIA |
---|---|---|
q2 | 0.43 | 0.54 |
r2 | 0.94 | 0.94 |
s | 0.09 | 0.09 |
F | 78.32 | 78.69 |
PLS components | 6 | 6 |
Field contribution | ||
Steric | 0.474 | 0.100 |
Electrostatic | 0.526 | 0.428 |
Hydrophobic | 0.283 | |
Donor | 0.146 | |
Acceptor | 0.044 | |
Bootstrapping r2 (20 runs) | 0.96±0.01 | 0.96±0.01 |
Randomization q2 (20 runs) | 0.33 | 0.39 |
Cross-validation q2 (20 runs) | 0.44 | 0.50 |