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. Author manuscript; available in PMC: 2014 Oct 10.
Published in final edited form as: J Med Chem. 2013 Sep 19;56(19):10.1021/jm401184f. doi: 10.1021/jm401184f

Table 3.

Inhibition in vitro binding affinities (Ki, nM) of reference compounds toward α7-nAChR. The binding assay conditions are the same as those in the Table 2.

Compound α7-nAChR
MLA 2.91 ± 0.76 (n = 9)
2 20.4
3 38.0
4 3.3
5 0.30, 0.50