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. 2014 Jan;85(1):91–104. doi: 10.1124/mol.113.089482

TABLE 1.

A number of antiasthma and antiallergenics act as potent agonists of human GPR35a

PathHunter human GPR35a–β-arrestin-2 interaction assays were performed using a CHO–K1 cell line stably expressing human GPR35 and β-arrestin-2. Data are presented as the mean ± S.E.M. and are derived from three independent experiments.

Compound EC50
nM
Nedocromil sodium 970 ± 87.0
Cromolyn disodium 2980 ± 127
Bufrolin 2.93 ± 0.71
Lodoxamide 1.61 ± 0.42
Nivimedone sodium 1930 ± 348
Tranilast No response