Table 5.
compound | HCT-116 | MRSA inhibition |
---|---|---|
| ||
IC50 (μg/mL) | MIC (μg/mL) | |
Napyradiomycin 1 | 4.19 | 16 |
Napyradiomycin 2 | >20 | 64 |
Napyradiomycin 3 | >20 | >64 |
Napyradiomycin 4 | 16.1 | >64 |
Napyradiomycin 5 | 4.81 | >64 |
Napyradiomycin 6 | 9.42 | >64 |
Napyradiomycin B2 (7) | 3.18 | 32–64 |
Napyradiomycin B3 (8) | 0.19 | 2 |
Napyradiomycin B4 (9) | 1.41 | 32 |