Table 1. Summary of Analogues and Antagonist Activity at TRPM2f.
See ref (21).
No significant inhibition at 100 μM; compounds were not evaluated further.
Antagonistic effect observed but not statistically significant; see relevant figure.
Could only be tested at 100 μM due to solubility difficulties.
Partial inhibition was observed at 900 μM; not evaluated further.
n.d. = not determined. n.s. = no significant antagonist effect observed.