Table 1. Summary of Analogues and Antagonist Activity at TRPM2^f.

^aSee ref (21).

^bNo significant inhibition at 100 μM; compounds were not evaluated further.

^cAntagonistic effect observed but not statistically significant; see relevant figure.

^dCould only be tested at 100 μM due to solubility difficulties.

^ePartial inhibition was observed at 900 μM; not evaluated further.

^fn.d. = not determined. n.s. = no significant antagonist effect observed.