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. Author manuscript; available in PMC: 2014 May 1.
Published in final edited form as: Biochim Biophys Acta. 2013 Jan 2;1827(5):10.1016/j.bbabio.2012.12.007. doi: 10.1016/j.bbabio.2012.12.007

Table 2.

Complex II modulators.

Reagent Conc. Effects mKATP effect
ATP mM Activate [102,162] Inhibit [102,182,198]
Atpenin A5 nM Inhibit [104,114,173,174] Activate [104]
Diazoxide μM Inhibit [171] Activate [102,115,182,198]
HNO μM Inhibit [108,109] Activate [108]
LNO2 μM Inhibit [108] Activate [108]
Malonate mM Inhibit [137] Activate [102,104,137,181]
3-nitropropionate mM Inhibit [236,237] Activate [113,137]
Oxaloacetate μM Inhibit [52,102,238,239]
Harzianopyridone nM Inhibit [114]
carboxin μM Inhibit [114]
HQNO μM Inhibit [114]
TTFA μM Inhibit [114]

Legend. HQNO, 2-heptyl-4-hydroxyquinoline N-oxide; TTFA, 4,4,4-trifluoro-1-(2-thienyl)-1,3-butanedione