Table 1.
Receptors | Endogenous ligands | Synthetic agonists | Synthetic antagonists |
---|---|---|---|
PPARα | LTB4 | Gemfibrozil | GW-6471 |
8-HETE | Fenofibrate | ||
Ciprofibrate | |||
Wy-14643 | |||
PPARβ/δ | 15-HETE | GW-0742 | GSK-0660 |
GW-501516 | GSK-3787 | ||
L-165041 | |||
PPARγ | 15d-PGJ2 | Rosiglitazone | GW-9662 |
15-HETE | Pioglitazone | ||
9-HODE | Troglitazone | ||
13-HODE | Ciglitazone |