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. 2012 Feb 28;33(3):217–222. doi: 10.1007/s10059-012-2297-y

Table 1.

Ligands for PPAR subfamily

Receptors Endogenous ligands Synthetic agonists Synthetic antagonists
PPARα LTB4 Gemfibrozil GW-6471
8-HETE Fenofibrate
Ciprofibrate
Wy-14643
PPARβ/δ 15-HETE GW-0742 GSK-0660
GW-501516 GSK-3787
L-165041
PPARγ 15d-PGJ2 Rosiglitazone GW-9662
15-HETE Pioglitazone
9-HODE Troglitazone
13-HODE Ciglitazone