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. 2013 Dec 17;170(8):1459–1581. doi: 10.1111/bph.12445
Nomenclature CT receptor AMY1 receptor AMY2 receptor AMY3 receptor
HGNC, UniProt CALCR, P30988
Subunits RAMP1 (Accessory protein), CT receptor RAMP2 (Accessory protein), CT receptor RAMP3 (Accessory protein), CT receptor
Principal transduction Gs Gs Gs Gs
Rank order of potency CT (salmon) ≥ CT ≥ AMY, α-CGRP > AM, AM2/IMD CT (salmon) ≥ AMY ≥ α-CGRP > AM2/IMD ≥ CT > AM Poorly defined CT (salmon) ≥ AMY > α-CGRP ≥ AM2/IMD ≥ CT > AM
Endogenous agonists (pKi) CT (Selective) (pEC50 9.0 – 11.2) 486,487,492,498,499,503 AMY AMY AMY
Radioligands (Kd) [125I]CT (salmon) (Agonist, Full agonist) (1x10−10 M), [125I]CT (human) (Agonist, Full agonist) (1x10−10 – 1x10−9 M) [125I]BH-AMY (rat, mouse) (Agonist, Full agonist) (1x10−10 – 1x10−9 M) [125I]BH-AMY (rat, mouse) (Agonist, Full agonist) (1x10−10 – 1x10−9 M) [125I]BH-AMY (rat, mouse) (Agonist, Full agonist) (1x10−10 – 1x10−9 M)