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. 2013 Dec 17;170(8):1459–1581. doi: 10.1111/bph.12445
Nomenclature HGNC, UniProt Principal transduction Selective agonists (pKi) Selective antagonists (pKi) Radioligands (Kd)
GPER GPER1, Q99527 Gs 761, Gi/o 763 G-1 (8.0) 757 G36 (pIC50 6.78–6.95) 760, G15 (pIC50 6.7) 759 [3H]17β-estradiol (Agonist, Full agonist) (2.7x10−9–3.3x10−9 M) 764