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. 2013 Dec 17;170(8):1459–1581. doi: 10.1111/bph.12445
Nomenclature HGNC, UniProt Principal transduction Rank order of potency Selective antagonists (pKi) Radioligands (Kd)
ghrelin receptor GHSR, Q92847 Gq/11 ghrelin = [des-Gln14]ghrelin 896,907 GSK1614343 (pKB 8.0 - Rat) 911, YIL781 (pKB 8.0) 899, GSK1614343 (pIC50 8.4) 912 [125I][His9]ghrelin (human) (Agonist, Full agonist) (4x10-10 M) 905, [125I][Tyr4]ghrelin (human) (Agonist, Full agonist) (4x10-10 M) 909