Nomenclature | HGNC, UniProt | Principal transduction | Rank order of potency | Selective antagonists (pKi) | Radioligands (Kd) |
ghrelin receptor | GHSR, Q92847 | Gq/11 | ghrelin = [des-Gln14]ghrelin 896,907 | GSK1614343 (pKB 8.0 - Rat) 911, YIL781 (pKB 8.0) 899, GSK1614343 (pIC50 8.4) 912 | [125I][His9]ghrelin (human) (Agonist, Full agonist) (4x10-10 M) 905, [125I][Tyr4]ghrelin (human) (Agonist, Full agonist) (4x10-10 M) 909 |