| Nomenclature | HGNC, UniProt | Principal transduction | Endogenous agonists (pKi) | Selective agonists (pKi) | Selective antagonists (pKi) | Radioligands (Kd) |
| kisspeptin receptor | KISS1R, Q969F8 | Gq/11 1048,1050 | kisspeptin-10 (Selective) (8.6–10.4) 1048,1051, kisspeptin-54 (Selective) (8.8–9.5) 1048,1051, kisspeptin-13 (Selective) (8.4) 1048 | 4-fluorobenzoyl-FGLRW-NH2 (pEC50 9.2) 1053, [dY]1KP-10 (pIC50 8.4 - Mouse) 1046 | peptide 234 1052 | [125I]kisspeptin-14 (human) 1049, [125I]Tyr45-kisspeptin-15 (Agonist, Full agonist) (1 × 10−10 M) 1051, [125I]kisspeptin-13 (human) (Agonist, Full agonist) (2 × 10−10 M) 1049, [125I]kisspeptin-10 (human) (Agonist, Full agonist) (1.9 × 10−9 M) 1048 |
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