Nomenclature | NTS1 receptor | NTS2 receptor |
HGNC, UniProt | NTSR1, P30989 | NTSR2, O95665 |
Principal transduction | Gq/11 | Gq/11 |
Rank order of potency | neurotensin > neuromedin N 1332 | neurotensin = neuromedin N 1335 |
Selective agonists (pKi) | JMV449 1338 | levocabastine (6.8) 1335,1337 |
Selective antagonists (pKi) | SR48692 (pIC50 7.5–8.2) 1331 | – |
Radioligands (Kd) | [3H]SR48692 (Antagonist) (3.2x10−9 M – Rat) 1333 | – |