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. 2013 Dec 17;170(8):1706–1796. doi: 10.1111/bph.12450
Nomenclature Organic cation transporter 1 Organic cation transporter 2 Organic cation transporter 3
Systematic nomenclature SLC22A1 SLC22A2 SLC22A3
Common abbreviation OCT1 OCT2 OCT3
HGNC, UniProt SLC22A1, O15245 SLC22A2, O15244 SLC22A3, O75751
Endogenous substrates 5-HT, PGE2, PGF2α, choline dopamine 303, histamine 303, PGE2 304 5-HT 307, (-)-noradrenaline 307, dopamine 307
Substrates tetraethylammonium, desipramine, MPP+, metformin, acyclovir (+)-tubocurarine 302, tetraethylammonium 302, pancuronium 302, MPP+ 302 quinidine, tetraethylammonium, MPP+
Stoichiometry Unknown Unknown Unknown