Nomenclature |
Organic cation transporter 1 |
Organic cation transporter 2 |
Organic cation transporter 3 |
Systematic nomenclature |
SLC22A1 |
SLC22A2 |
SLC22A3 |
Common abbreviation |
OCT1 |
OCT2 |
OCT3 |
HGNC, UniProt |
SLC22A1, O15245
|
SLC22A2, O15244
|
SLC22A3, O75751
|
Endogenous substrates |
5-HT, PGE2, PGF2α, choline |
dopamine 303, histamine 303, PGE2 304
|
5-HT 307, (-)-noradrenaline 307, dopamine 307
|
Substrates |
tetraethylammonium, desipramine, MPP+, metformin, acyclovir |
(+)-tubocurarine 302, tetraethylammonium 302, pancuronium 302, MPP+ 302
|
quinidine, tetraethylammonium, MPP+ |
Stoichiometry |
Unknown |
Unknown |
Unknown |