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. 2013 Dec 17;170(8):1797–1867. doi: 10.1111/bph.12451
Nomenclature Diacylglycerol lipase α Diacylglycerol lipase β N-Acylphosphatidylethanolamine-phospholipase D
Common abbreviation DGLα DGLβ NAPE-PLD
HGNC, UniProt DAGLA, Q9Y4D2 DAGLB, Q8NCG7 NAPEPLD, Q6IQ20
EC number 3.1.1.- 3.1.1.-
Selective inhibitors (pIC50) RHC80267, orlistat (7.2) 196 RHC80267, orlistat (7.0) 196
Comment NAPE-PLD activity appears to be enhanced by polyamines in the physiological range 202, but fails to transphosphatidylate with alcohols 205 unlike phosphatidylcholine-specific phospholipase D