Table 6.

Biological activity of anilinoalcohols with varying substitutions on ring I

Compound	Ring II (meta or para)	R	Percent inhibition of anilinoalcohol	Percent inhibition of corresponding ketone
95	p	H	33%	4%
96	m	H	4%	32%
97	p	p-CH3	15%	12%
98	m	p-CH3	8%	7%
99	m	m-CH3	3%	38%
100	p	p-Cl	27%	2%
101	m	p-Cl	0%	24%
102	p	m-Cl	20%	0%
103	m	m-Cl	23%	0%
104	p	p-OMe	26%	0%
105	m	p-OMe	14%	2%
106	p	m-OMe	32%	14%
107	m	m-OMe	24%	9%
108	m	p-COCH3	19%	6%
109	p	m-COCH3	22%	18%
110	p	p-COOCH2CH3	22%	9%