Table 3.
Effects of homologation and transposition of linker chain on SOICR inhibition.
| entry | compound | structure | IC50 (μM) ± SEM | repeats (n) | no. of cells |
|---|---|---|---|---|---|
| 1 | 2 |
|
16.8 ± 3.3 | 4 | 206 |
| 2 | 32 |
|
14.6 ± 3.5 | 3 | 177 |
| 3 | 33 |
|
11.4 ± 0.8 | 3 | 245 |
| 4 | 34 |
|
13.5 ± 2.3 | 3 | 163 |
| 5 | 35 |
|
86.7 ± 53 | 3 | 204 |
| 6 | 36 |
|
20.0 ± 1.6 | 3 | 167 |
| 7 | 37 |
|
10.2 ± 0.5 | 3 | 168 |
| 8 | 38 |
|
9.51 ± 2.3 | 3 | 217 |
| 9 | 39 |
|
24.4 ± 3.1 | 4 | 365 |
| 10 | 40 |
|
26.7 ± 3.2 | 7 | 381 |