Table 3.
Concentrations
|
AUC0–16ha
|
t1/2b
|
||||
---|---|---|---|---|---|---|
MPE%c | MAPE%d | MPE%c | MAPE%d | MPE%c | MAPE%d | |
Plasma | 28.53 | 43.36 | 16.18 | 16.18 | 9.57 | 12.64 |
Intestine | −8.40 | 68.10 | 9.77 | −9.77 | 6.09 | 6.09 |
Liver | 23.57 | 51.03 | 4.10 | −1.70 | 19.11 | 19.11 |
Kidney | 45.40 | 52.90 | 8.11 | 8.11 | 18.57 | 18.57 |
Heart | 52.81 | 73.34 | 18.33 | 13.18 | 15.41 | 15.41 |
Lung | 4.45 | 59.25 | 24.22 | −1.79 | 25.14 | 25.14 |
Slowly perfused | 28.77 | 47.40 | 27.99 | −4.53 | 16.24 | 22.96 |
Brain | 53.30 | 63.65 | 7.30 | 6.24 | −4.29 | 19.16 |
AUC0–16 h is the area under the concentration–time curve from 0 to 16 h
t1/2 is the half-life for elimination as calculated from linear regression of the terminal elimination phase
MPE% is the median prediction error, which is a measure of the bias of the prediction
MAPE% is the median absolute prediction error, which is a measure of the precision of the prediction