Table 1. The association schemes of MDM2 interaction with Nutlin-3 geometrical isomers.
Protein | Ligand | Complex | Scheme | |
---|---|---|---|---|
MDM2 + | Nutlin-3a | → | MDM2:Nutlin-3a | (1) |
Nutlin-3b | → | MDM2:Nutlin-3b | ||
MDM2 + | trans-Nutlin-3a | → | MDM2:trans-Nutlin-3a | (2) |
trans-Nutlin-3b | → | MDM2:trans-Nutlin-3b |