Table 1. Structure of glutaminase inhibitors employed [17].
Compound | Molecular Structure | Glutaminase activity (IC50, μM) |
---|---|---|
BPTES |
![]() |
3 |
JHU-198 |
![]() |
4 |
JHU-212 |
![]() |
30 |
JHU-329 |
![]() |
>100 |
Compound | Molecular Structure | Glutaminase activity (IC50, μM) |
---|---|---|
BPTES |
![]() |
3 |
JHU-198 |
![]() |
4 |
JHU-212 |
![]() |
30 |
JHU-329 |
![]() |
>100 |