Skip to main content
. Author manuscript; available in PMC: 2014 Feb 24.
Published in final edited form as: Exp Biol Med (Maywood). 2011 May 12;236(6):637–647. doi: 10.1258/ebm.2011.010389

Table 1.

List of CXCR4 inhibitors, their chemical structures, sequences and modifications

Inhibitors Modification diagrams or chemical structures Amino acid sequences* References
ALX40-4C AcNH-D-Arg-(D-Arg)8-COOH 55,93,94
AMD3100 graphic file with name nihms544753t1.jpg 82
CGP64222 graphic file with name nihms544753t2.jpg 97
R3G graphic file with name nihms544753t3.jpg 97
T22 graphic file with name nihms544753t4.jpg RRWCYRKCYKGYCYRKCR 83
T140 graphic file with name nihms544753t5.jpg R-R-Na1-C-Y-R-K-D(K)-P-Y-R-Cit-C-R 95,96
TC14012 graphic file with name nihms544753t6.jpg R-R-Na1-C-Y-Cit-K-D(Cit)-P-Y-R-Cit-C-R 95
FC131 graphic file with name nihms544753t7.jpg 96
SDF-1α graphic file with name nihms544753t8.jpg KPVSLSYRCPCRFFESHVARANVKHLKILNTPNCALQIVARLKNNNRQVCIDPKLKWIQEYLEKALNK 1,6,7,58,84,85,91
vMIP-II graphic file with name nihms544753t9.jpg LGASWHRPDKCCLGYQKRPLPQVLLSSWYPTSQLCSKPGVIFLTKRGRQVCADKSKDWVKKLMQQLPVTAR 8,9,31
V1 graphic file with name nihms544753t10.jpg LGASWHRPDKCCLGYQKRPLP 38
DV1 graphic file with name nihms544753t11.jpg LGASWHRPDKCCLGYQKRPLP 39
RCP168 graphic file with name nihms544753t12.jpg LGASWHRPDKCCLGYQKRPLPQVLLSSWYPTSQLCSKPGVIFLTKRGRQVCADKSKDWVKKLMQQLPVTAR 72
*

D-Amino acids are shown in italic