Table 1.
C-027 Pharmacokinetics in mice
Dose (mg/kg) | Route | Cmax (ng/mL) | Tmax (hr) | AUC0-last (hr * ng per mL) | Vss (L/kg) | F* (%) |
---|---|---|---|---|---|---|
5 | i.v. | 1424 | 0.083 | 302 | 37.1# | ND |
1 | i.p. | 12.9 | 0.5 | 21.5 | ND | ND |
10 | i.p | 333 | 0.5 | 363 | ND | ND |
10 | o.g. | 22.7 | 2 | 134 | ND | 22 |
Bioavailability.
Represents ~63 × the total body water volume.
C-027 was administered to CD-1 mice either via i.v., i.p., or o.g. routes at various concentrations. The peak concentration (Cmax) and time of Cmax (Tmax) were token directly from the observed data. The AUC, apparent volume of distribution (Vss), and bioavailability (F) were estimated with the linear trapezoidal rule using WinNonlin software Version 4.2 (Pharsight, Mountain View, CA).
AUC = area under the curve; i.v. = intravenous; i.p. = intraperitoneal; o.g. = oral lavage.