Table 2. Yield of Heterocycle-Forming MCR with Different Isocyanides.
entry | R1 | yield [%] |
---|---|---|
1 | cyclohexyl | 70 |
2 | 4-OMe-Ph | 100 |
3 | 4-F-Ph | 28 |
4 | naphth-2-yl | 59 |
5 | tBu | 90 |
6 | 1-adamantyl | 61 |
7 | 2,6-diMe-Ph | 0 |
entry | R1 | yield [%] |
---|---|---|
1 | cyclohexyl | 70 |
2 | 4-OMe-Ph | 100 |
3 | 4-F-Ph | 28 |
4 | naphth-2-yl | 59 |
5 | tBu | 90 |
6 | 1-adamantyl | 61 |
7 | 2,6-diMe-Ph | 0 |