Table 2.
IC50/IC25 (nmol/L) | ||||||||
---|---|---|---|---|---|---|---|---|
Drug | C-TAC | CML-1 | CML-6M | CMT-12 | CMT-27 | DEN-HSA | Abrams | D17 |
343074 | 19.0/10.4 | 51.4/7.3 | 55.3/5.1 | 4.6/2.0 | 3.7/1.7 | 180.0/56.4 | 6.4/2.8 | 10.0/5.3 |
424044 | NA/NA | 78.6/22.8 | 61.6/24.0 | 78.8/42.6 | 35.6/21.5 | NA/NA | 104.1/73.3 | 10.7/4.4 |
NA, not achieved.
GS analogue was administered to cells in MEM supplemented with 10% (C/10) FBS.