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Concentration-dependence of hMGL Inhibition by AM6701 and NAM
| Inhibitor | Inhibitor:hMGL molar ratio |
hMGL Inhibition (%) 10 min |
|---|---|---|
| AM6701 | 1:1 | 72 |
| 3.3:1 | 85 | |
| 8.3:1 | 91 | |
| NAM | 1:1 | 51 |
| 3.3:1 | 80 | |
| 8.3:1 | 82 | |
| 33:1 | 84 |
Reporter substrate (AHMMCE) concentration was 50 μM.
