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. Author manuscript; available in PMC: 2015 Mar 25.
Published in final edited form as: Chem Commun (Camb). 2014 Feb 12;50(24):3151–3154. doi: 10.1039/c4cc00394b

Table 1.

Results of the screening of various ynamide nucleophiles.a

graphic file with name nihms-568450-t0005.jpg
Entry Ynamide Product Time
(h)
Yielda
(%)
Ee
(%)
1 graphic file with name nihms-568450-t0006.jpg graphic file with name nihms-568450-t0007.jpg 2.5 87 60
2 graphic file with name nihms-568450-t0008.jpg graphic file with name nihms-568450-t0009.jpg 3 91 38
3 graphic file with name nihms-568450-t0010.jpg graphic file with name nihms-568450-t0011.jpg 5 100 27
4 graphic file with name nihms-568450-t0012.jpg graphic file with name nihms-568450-t0013.jpg 18 68 80
5 graphic file with name nihms-568450-t0014.jpg graphic file with name nihms-568450-t0015.jpg 18 58 78
6 graphic file with name nihms-568450-t0016.jpg graphic file with name nihms-568450-t0017.jpg 24 87 77
7 graphic file with name nihms-568450-t0018.jpg graphic file with name nihms-568450-t0019.jpg 27 60 81
a

Based on NMR analysis