Table 1.
Cell Line | Mutational Status | PP242 (μM) | ||
---|---|---|---|---|
KRAS | PIK3CA | bRAF | ||
SW620 | G12V | WT | WT | 7.8 |
SW480 | G12V | WT | WT | 4.6 |
SK-CO-1 | G12V | WT | WT | 4 |
LS-513 | G12D | WT | WT | 3.9 |
SW1116 | G12A | WT | WT | 0.84 |
LS-174T | G12D | H1047R | WT | 0.84 |
HCT 116 | G13D | H1047R | WT | 0.41 |
HCT 15 | G13D | E545K | WT | 0.3 |
COLO 205 | WT | WT | V600E | 0.24 |
HT-29 | WT | WT | V600E | 0.23 |
COLO 201 | WT | WT | V600E | 0.23 |
Caco-2 | WT | WT | WT | 0.22 |
SW48 | WT | WT | WT | 0.09 |