Figure 1.
(A) Repression of p21 gene transcription by HDAC1/2. p21 inhibits the cyclin-cdk complex at the indicated phases (G1/S, S, and G2/M) to block cell cycle progression. HDAC1/2 binds to Sp1/Sp3 and is recruited to the promoter site of p21, leading to hypoacetylation of the promoter region and inhibition of p21 transcription. (B) Repression of p21 gene transcription by HDAC3/4. HDAC3/4 is recruited to the promoter site by binding to the Sp1/3 transcription factor as part of a larger repressor complex, NCo-R-SMRT, to inhibit p21 transcription.