TABLE 2.
OSIP108 or analogue | Peptide | BIC-2 (μM) | Fold change |
---|---|---|---|
OSIP108 | MLCVLQGLRE | 5.3 | |
S-OSIP108 | ELRLVCMGQL | >100 | >20 |
d-OSIP108 | MLCVLQGLRE (all d-amino acids) | 13.7 | 2.6 |
[CYC1]OSIP108 | Cyclo-MLCVLQGLRE | >100 | >20 |
[CYC2]OSIP108 | Cyclo-MLCVLQGLREGG | 36.0 | 6.8 |
[CYC3]OSIP108 | Cyclo-MLCVLQGLREC | >100 | >20 |