TABLE 2.
Significant steps in piperacillin-tazobactam population plasma PK model-building processa
Population model | OFV | ΔOFVb |
---|---|---|
Piperacillin | ||
V = θV · WT | 1,125 | |
CL = θCL · WT | 1,125 | |
CL = θCL · WT · (PMA/33)COVPMA | 1,113 | −12 |
CL = θCL · WT · (SCR/0.5)COVSCR | 1,106 | −19 |
CL = θCL · WT · (SCR/0.5)COVSCR · COVGENTGENT | 1,093 | −13 |
CL = θCL · WT · (SCR/0.5)COVSCR · COVGENTGENT · (PMA/33)COVPMA | 1,092 | −1 |
Tazobactam | ||
V = θV · WT | 509 | |
CL = θCL · WT | 509 | |
CL = θCL · WT · (PMA/33)COVPMA | 491 | −18 |
CL = θCL · WT · (SCR/0.5)COVSCR | 491 | −18 |
CL = θCL · WT · (SCR/0.5)COVSCR · COVGENTGENT | 480 | −11 |
CL = θCL · WT · (SCR/0.5)COVSCR · COVGENTGENT · (PMA/33)COVPMA | 470 | −10 |
WT, actual body weight (kg); SCR, serum creatinine (mg/dl); GENT = 1 if gentamicin was given concurrently with piperacillin-tazobactam, and GENT = 0 if there was no concurrent therapy; PMA, postmenstrual age (weeks); OFV, objective function value.
For multivariable models, the change in OFV is relative to the prior model.