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. Author manuscript; available in PMC: 2015 Mar 20.
Published in final edited form as: Brain Res. 2014 Jan 25;1554:36–48. doi: 10.1016/j.brainres.2014.01.036

Table 1.

Binding affinity (Ki, nM) of SH-I-048A and diazepam at human recombinant GABAA receptors containing β3, γ2 and named α subunit, stably expressed in mouse fibroblast L(tk−) cells; ND – not detected. [3H] flunitrazepam was used as the radiolabelled ligand in the competition binding assay. Data for diazepam were published in Savić et al. 2010.

Ligand α1 α2 α3 α4 α5 α6
SH-I-048A 0.77 0.17 0.38 ND 0.11 ND
diazepam 14.0 7.8 13.9 ND 13.4 ND