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Binding affinity (Ki, nM) of SH-I-048A and diazepam at human recombinant GABAA receptors containing β3, γ2 and named α subunit, stably expressed in mouse fibroblast L(tk−) cells; ND – not detected. [3H] flunitrazepam was used as the radiolabelled ligand in the competition binding assay. Data for diazepam were published in Savić et al. 2010.