Table 2. Autophagy inhibitors.
| Name | Mechanism | Target point | Solubility | References |
|---|---|---|---|---|
| 3-Methyladenine | PI 3-kinase inhibitor | Autophagosome formation | Water-soluble | 76,78,80 |
| Wortmaninn | PI 3-kinase inhibitor | Autophagosome formation | Water-insoluble | 80,102,103 |
| LY294002 | PI 3-kinase inhibitor | Autophagosome formation | Water-insoluble | 80,102,103 |
| Cycloheximide | protein synthesis inhibitor | Autophagosome formation | Water-insoluble | 85,86,87 |
| Bafilomycin A1 | Vacuolar-type H(+)-ATPase inhibitor | Autophagolysosome formation | Water-insoluble | 90,91 |
| Hydroxychloroquine | Lysosomal lumen alkalizer | Lysosome | Water-soluble | 95,104,105 |
| Lys05 | Lysosomal lumen alkalizer | Lysosome | Water-soluble | 97,106 |
| Leupeptin | Acid protease inhibitor | Lysosome | Water-soluble | 98,107 |
| E64d | Acid protease inhibitor | Lysosome | Water-insoluble | 100,108 |
| Pepstatin A | Acid protease inhibitor | Lysosome | Water-insoluble | 100 |