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. 2013 Jul 29;34(9):1149–1155. doi: 10.1038/aps.2013.66

Table 2. Effects of SKF83959 and DOV21947 on the transporting kinetics of SERT, NET, and DAT.

		Compound
		Vehicle	DOV21947	SKF83959
SERT	V_max (cpm/min·10⁶ cells)	6581±305	7216±732	7426±580
	K_t (nmol/L)	104.50±21.09	362.20±23.32^b	316.70±64.13^b
	K_i (μmol/L)	–	0.89±0.24	1.43±0.45
NET	V_max (cpm/min·10⁶ cells)	246.30±23.61	40.70±9.00^b	104.5±11.05^be
	K_t (nmol/L)	13.24±3.13	13.69±2.21	13.30±2.19
	K_i (μmol/L)	–	0.18±0.04	0.60±0.08^e
DAT	V_max (cpm/min·10⁶ cells)	224.00±14.6	265.20±29.29	116.00±7.45^b
	K_t (nmol/L)	29.65±4.73	68.05±14.11^b	30.81±3.37
	K_i (μmol/L)	–	1.47±0.31	9.01±0.80^e

The parameters were obtained from Figure 2. Data were expressed as mean±SEM. ^bP<0.05 vs vehicle. ^eP<0.05 vs DOV21947.