Effects of Aβ oligomers on the activation
of caspase-3. The
NucView488 substrate used to monitor the activation of caspase-3 in
real time becomes fluorescent when cleaved by caspase-3 and subsequently
migrates to the nucleus. The kinetics of caspase-3 activation were,
therefore, monitored by measuring the fluorescence within each cell
as a function of time. In the kinetic traces shown here, each line
represents a single cell with data for neurons in red and for astrocytes
in black. Additionally, end point measurements of net caspase-3 activation
after 30 min of observation were taken by counting the number of cells
observed with fluorescent nuclei as a fraction of total cells observed.
The experiments were performed on at least 4 different samples. (A)
Fluorescence of the NucView488 caspase-3 substrate as a function of
time following treatment of primary cultures containing both neurons
and astrocytes with 500 nM Aβ42 (containing 19.5 nM oligomers);
370 cells were monitored over 6 samples. (B) Fluorescence of the NucView488
caspase-3 substrate as a function of time following the treatment
of primary cultures containing both neurons and astrocytes with 500
nM of monomeric Aβ42; 187 cells were monitored over 4 samples.
(C) Proportion of cells (%) that experience activation of caspase-3
following 30 min of incubation with monomeric Aβ42 (500 nM)
or oligomeric Aβ42 solutions (total peptide concentrations of
50 nM and 500 nM with oligomer concentrations of 1.95 nM and 19.5
nM). These data are the end points (after 30 min) of experiments presented
in A and B. For experiments using 50 nM of Aβ42, 231 cells were
monitored over 4 different samples. ** signifies a p-value <0.01 by a Mann–Whitney nonparametric rank correlation.
Comparisons were performed relative to the data obtained with 500
nM of Aβ42 oligomers. (D) Fluorescence of the NucView488 caspase-3
substrate as a function of time following the treatment of primary
hippocampal cultures containing both neurons and astrocytes with 500
nM Aβ42 (containing 19.5 nM oligomers). Cultures in this experiment
had been pretreated with the NADPH-oxidase inhibitor, AEBSF (20 μM),
for 30 min prior to the addition of Aβ42; 154 cells were monitored
in a single sample. (E) Fluorescence of the NucView488 caspase-3 substrate
as a function of time following the treatment of primary hippocampal
cultures containing both neurons and astrocytes with 500 nM Aβ42
(containing 19.5 nM oligomers). The cultures in this experiment had
been pretreated with the NADPH-oxidase inhibitor, DPI (0.5 μM),
for 30 min prior to the addition of Aβ42; 138 cells were monitored
on a single sample. Control experiments to verify that the observed
effects on caspase-3 activation are not affected by the fluorophores
attached to the Aβ peptides are reported in Figure S2E,F, Supporting Information.