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. Author manuscript; available in PMC: 2014 May 1.
Published in final edited form as: Curr Top Med Chem. 2013;13(7):813–820. doi: 10.2174/1568026611313070004

Table 1.

Correlations on the different data sets used between experimental and predicted Vu,brain values provided by our physical model.

# Compounds Reference Type of data R2
52 Friden 2011 Slice 0.70
33 Maurer 2005 Homogenate 0.69
12 Becker 2006 + Ooie 1997 Slice, Microdialysis 0.79
34 Kalvass 2007 Homogenate 0.32
15 Summerfield 2006 Homogenate 0.13
146 All data sets Slice, Homogenate 0.55