Table 2. Selectivity of 7Fb and 7Fc for a panel of protein phosphatases.
|
|
|
|
IC50 (μmol/L) |
|
|
---|---|---|---|---|---|---|
Compd | PTP1B | LAR | Cdc25B | SHP1 | SHP2 | PRL3 |
7Fb | 0.69±0.07 | >50 | 2.22±0.14 | >50 | >50 | 5.34±1.42 |
7Fc | 0.48±0.07 | >50 | 0.89±0.03 | 1.90±0.17 | 1.61±0.13 | 2.07±0.50 |