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| FLIPR | binding |
|||
|---|---|---|---|---|
| compd | stereo | human EC50 (μM)a | human Ki (μM)b | rat Ki (μM)b |
| 9a | S | 0.014 | 0.038 | 0.14 |
| 9b | R | 0.37 | 1.6 | |
The activity was measured with anhydrous 9a. The value is an average of n = 3 in the presence of 0.1% BSA.
All values are averages of n = 2 or 3 in the presence of 0.2% BSA.
